ICVAA - Betablockers II

 


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Angiotensin-converting enzyme inhibitors (ACE inhibitors): are indicated for heart failure, diabetes, recurrent stroke prevention, postmyocardial infarction, people at high risk for coronary disease,and chronic kidney disease.  benazepril (Lotensin), captopril (Capoten), enalapril (Vasotec), fosinopril (Monopril), lisinopril (Prinivil, Zestril), moexipril (Univasc), quinapril (Accupril), ramipril (Altace), and trandolapril (Mavik).

KNOW:  ACE inhibitors have been shown to decrease morbidity and mortality in patients with heart failure and are first line treatment for heart failure.  Additionally, ACE inhibitors are indicated for diabetics type 1 with nephropathy, patients with proteinuria greater than 1 gram per 24 hours, and patients with renal insufficiency.  These drugs should be used cautiously in patients with a creatinine greater than or equal to 3 mg/dl and/or patients with renovascular disease. 

KNOW:  ACE inhibitors are contraindicated in pregnancy.  ACE inhibitors are associated with a cough in some patients that resolves when the drug is discontinued.  Hyperkalemia can occur in patients taking an ACE inhibitor especially if the patient is also taking a potassium-sparing diuretic or a potent NSAID.  Angioedema, neutropenia, and rashes are rare side effects of ACE inhibitors.  Patients with a history of angioedema should avoid ACE inhibitors.

-ACE inhibitors should be used with caution in patients with renovascular disease such as bilateral renal artery stenosis, and in patients with one kidney and unilateral renal artery stenosis since they may produce or worsen renal insufficiency.

-Captopril has the shortest half-life of the ACE inhibitors. 

-Enalapril has an IV form called enalaprilat which is the only ACE inhibitor that can be given IV.

Angiotensin II receptor blockers (ARB):  candesartan (Atacand), losartan (Cozaar), irbesartan (Avapro), and  valsartan (Diovan). These drugs are alternative agents to treat heart failure in patients who develop a cough while taking ACE inhibitors.  Other indications for ARB are diabetes and chronic kidney disease.  

KNOW:  angiotensin II receptor blockers are contraindicated in pregnancy. 

In general, angiotension II receptor blockers have the same contraindication and precautions as ACE inhibitors.

 

 
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